发明名称 CRYSTALLINE SOLIFENACIN SUCCINATE
摘要 <p>Crystalline solifenacin succinate, the solifenacin succinate having an average axial ratio of 5:1 or less, preferably an average axial ratio of 5:1 to 1:1, more preferably an average axial ratio of 1:1, and having at least one of the following properties: a) a particle size d 0.9 < 200 µm; b) an average particle size of approximately 2 to 40 µm; and c) peaks in the X-ray powder diffractogram at 3.7; 11.1; 18.6; 21.8° 2? ± 0.2° 2?.</p>
申请公布号 EP2638039(A1) 申请公布日期 2013.09.18
申请号 EP20110782419 申请日期 2011.11.11
申请人 HEXAL AG 发明人 BORN, MAX
分类号 C07D453/02;A61K31/472;A61P13/00 主分类号 C07D453/02
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