发明名称 NEW QUINAZOLINE COMPOUND
摘要 PROBLEM TO BE SOLVED: To provide a quinazoline compound having a GPR119 receptor agonistic activity and being useful as a medicine.SOLUTION: A compound expressed by general formula [I] or a pharmacologically acceptable salt thereof is provided. [In formula, Rrepresents hydrogen or halogen; ring A represents a 5- or 6-membered aryl ring (the aryl ring may contain one to four heteroatoms which are selected from O, S and N, and are the same or different); Rand Reach independently represents a halogen atom, a cyano group or the like; ring B represents a 6- or 7-membered aliphatic nitrogen-containing heterocyclic group; Rrepresents hydrogen or alkyl; Rrepresents hydrogen or a hydroxy group; and Rrepresents a hydroxy group, a cyano group or the like].
申请公布号 JP2013177321(A) 申请公布日期 2013.09.09
申请号 JP20100274645 申请日期 2010.12.09
申请人 MITSUBISHI TANABE PHARMA CORP 发明人 INOUE SHINYA;TSUBOI YASUNORI;IKEDA YOSUKE;NAKAJIMA TATSUO;FUJIMOTO NOBUAKI;IWASAKI SATOSHI;FUKANO YASUSHI
分类号 C07D239/94;A61K31/517;A61K31/5355;A61K31/5377;A61K31/551;A61P3/00;A61P3/04;A61P3/06;A61P3/10;A61P9/00;A61P9/10;A61P9/12;A61P43/00;C07D401/04;C07D401/14;C07D413/12;C07D413/14;C07D417/14 主分类号 C07D239/94
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