发明名称 |
SUBSTITUTED [(5H-PYRROLO[2,1-c] [1,4]BENZODIAZEPIN-11-YL)PIPERAZIN-1-YL]-2,2-DIMETHYLPROPANOIC ACID COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A< /sub> ANTAGONISTS. |
摘要 |
<p>A dual H1/5-HT2A receptor antagonist of the formula:, its uses, and methods for its preparation are described.</p> |
申请公布号 |
MX2013008786(A) |
申请公布日期 |
2013.09.06 |
申请号 |
MX20130008786 |
申请日期 |
2012.01.25 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
ANNE MARIE CAMP;PETER THADDEUS GALLAGHER;DAVID ANDREW COATES;ADAM JAN SANDERSON;ANDREW JAMES LEDGARD |
分类号 |
C07D487/04;A61K31/5517;A61P25/20 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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