发明名称 |
Compuestos derivados de carboxamidas azaheterociclicas biciclicas (quinazolinas), como inhibidores de quinasa p70s6k; proceso de preparacion; composicion farmaceutica; kit; y su uso para el tratamiento de enfermedades hiperproliferativas, tal como cancer, inflamacion, enfermedades relacionadas con vasculogenesis. |
摘要 |
The invention provides novel bicyclic azaheterocyclic carboxamide compounds according to Formula (I), their manufacture and use for the treatment of hyperproliferative diseases, such as cancer. |
申请公布号 |
CL2013000263(A1) |
申请公布日期 |
2013.09.06 |
申请号 |
CL20130000263 |
申请日期 |
2013.01.28 |
申请人 |
MERCK PATENT GMBH |
发明人 |
JONES REINALDO C;DESELM LIZBETH CELESTE;XIAO YUFANG;KARRA SRINIVASA R;LAN RUOXI;MOCHAKIN IGOR;SUTTON AMANDA E;RICHARDSON THOMAS E;HUCK BAYARD R;NEAGU CONSTANTIN |
分类号 |
C07D239/74;A61K31/517;A61P35/00;C07D403/12 |
主分类号 |
C07D239/74 |
代理机构 |
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地址 |
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