发明名称 PROCESS FOR THE PREPARATION OF ENANTIOMERIC FORMS OF 2,3-DIAMINOPROPIONIC ACLD DERIVATIVES
摘要 The disclosure relates to a process for the preparation of the enantiomeric forms of 2,3-diaminopropionic acid derivatives of formula I, wherein R1, R2 and R3 are defined as in the dsiclosure, by racemate resolution. The separation of the racemate into its enantiomers takes place through formation of diastereomeric salts upon addition of an enantiomerically pure auxiliary, and subsequent separation by fractional crystallization.
申请公布号 KR20130099044(A) 申请公布日期 2013.09.05
申请号 KR20137006179 申请日期 2011.08.05
申请人 SANOFI 发明人 GRAF CLAUS DIETER;RIEKE ZAPP JOERG
分类号 C07D239/42;A61K31/505 主分类号 C07D239/42
代理机构 代理人
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