Compounds having the formula I wherein A, Z, R1a, R1b, R2, R3, R4, R5, R6, R7, R9, R10, Ra, Rb and n are as defined herein are inhibitors of PAK1. Also disclosed are compositions and methods for treating cancer and hyperproliferative disorders.
申请公布号
US2013225620(A1)
申请公布日期
2013.08.29
申请号
US201213593776
申请日期
2012.08.24
申请人
ALIAGAS-MARTIN IGNACIO;CRAWFORD JAMES;LEE WENDY;MATHIEU SIMON;RUDOLPH JOACHIM;GENENTECH, INC.
发明人
ALIAGAS-MARTIN IGNACIO;CRAWFORD JAMES;LEE WENDY;MATHIEU SIMON;RUDOLPH JOACHIM