发明名称 PROCESSES FOR PREPARATION OF EVEROLIMUS AND INTERMEDIATES THEREOF
摘要 The present disclosure discloses processes of Everolimus and intermediates: reacting Sirolimus (Rapamycin) under solvent free conditions with appropriate side chain implying portion wise additions, one pot conversion, and resin mediated synthesis.
申请公布号 US2013225823(A1) 申请公布日期 2013.08.29
申请号 US201113988265 申请日期 2011.11.17
申请人 VENKATA SRINIVAS PULLELA;EKAMBARAM GANESH;KOTHAKONDA KIRAN KUMAR;PRASAD ANEGONDI SREENIVASA 发明人 VENKATA SRINIVAS PULLELA;EKAMBARAM GANESH;KOTHAKONDA KIRAN KUMAR;PRASAD ANEGONDI SREENIVASA
分类号 C07D498/16 主分类号 C07D498/16
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