发明名称 |
PROCESSES FOR PREPARATION OF EVEROLIMUS AND INTERMEDIATES THEREOF |
摘要 |
The present disclosure discloses processes of Everolimus and intermediates: reacting Sirolimus (Rapamycin) under solvent free conditions with appropriate side chain implying portion wise additions, one pot conversion, and resin mediated synthesis.
|
申请公布号 |
US2013225823(A1) |
申请公布日期 |
2013.08.29 |
申请号 |
US201113988265 |
申请日期 |
2011.11.17 |
申请人 |
VENKATA SRINIVAS PULLELA;EKAMBARAM GANESH;KOTHAKONDA KIRAN KUMAR;PRASAD ANEGONDI SREENIVASA |
发明人 |
VENKATA SRINIVAS PULLELA;EKAMBARAM GANESH;KOTHAKONDA KIRAN KUMAR;PRASAD ANEGONDI SREENIVASA |
分类号 |
C07D498/16 |
主分类号 |
C07D498/16 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|