发明名称 PYRAZOLO[1,5-a]PYRIMIDINE COMPOUNDS AS mTOR INHIBITORS
摘要 The present invention provides Pyrazolopyrimidine Compounds of Formula (I): wherein L, T, Z, U, V, W, R3, R6, R7, R8, and m are as defined herein, and pharmaceutically acceptable salts of such Pyrazolopyrimidine Compounds. The Pyrazolopyrimidine Compounds are useful in the treatment of cancer and other diseases or disorders wherein mTOR is deregulated.
申请公布号 EP2525659(A4) 申请公布日期 2013.08.28
申请号 EP20110735040 申请日期 2011.01.18
申请人 MERCK SHARP & DOHME CORP. 发明人 SIDDIQUI, M. ARSHAD;NAN, YANG;PATEL, MEHUL, F.;REDDY, PANDURANGA ADULLA P.;MANSOOR, UMAR FARUK;MENG, ZHAOYANG;VITHARANA, LALANTHI DILRUKSHI;ZHAO, LIANYUN;MANDAL, AMIT, K.;LIU, DUAN;TANG, SHUYI;MCRINER, ANDREW;BELANGER, DAVID, B.;CURRAN, PATRICK, J.;DAI, CHAOYANG;ANGELES, ANGIE, R.;YANG, LIPING;DANIELS, MATTHEW HERSH
分类号 A01N43/90 主分类号 A01N43/90
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