发明名称 |
Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors |
摘要 |
A process for the preparation of a compound of formula (I) comprising the steps: (a) reacting a compound of formula (II) wherein L and L' are suitable leaving groups, with a compound of formula (III) UNH2(III) to prepare a compound of formula (IV) and subsequently (b) substituting the group R1 by replacement of the leaving group L'.
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申请公布号 |
US8513262(B2) |
申请公布日期 |
2013.08.20 |
申请号 |
US20100691784 |
申请日期 |
2010.01.22 |
申请人 |
CARTER MALCOLM CLIVE;COCKERILL GEORGE STUART;LACKEY KAREN ELIZABETH;GLAXOSMITHKLINE LLC |
发明人 |
CARTER MALCOLM CLIVE;COCKERILL GEORGE STUART;LACKEY KAREN ELIZABETH |
分类号 |
A01N43/90;A61K31/47;A61K31/4709;A61K31/505;A61K31/517;A61K31/519;A61P9/10;A61P17/06;A61P29/00;A61P35/00;A61P43/00;C07D221/00;C07D239/00;C07D239/72;C07D239/94;C07D405/04;C07D405/14;C07D417/04;C07D417/14;C07D471/04 |
主分类号 |
A01N43/90 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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