发明名称 ANHYDROUS POLYMORPHS OF [(2R,3S,4R,5R)-5-(6-(CYCLOPENTYLAMINO)-9H-PURIN-9-YL)-3,4-DIHYDROXYTETRAHYDROFURAN-2-YL)} METHYL NITRATE AND PROCESSES OF PREPARATION THEREOF
摘要 <p>The present invention provides novel anhydrous polymorph forms of 2R,3S,4R,5R)-5-(6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl nitrate (Compound A). The present invention also provides processes for preparation of the anhydrous polymorphic forms of compound A.</p>
申请公布号 CA2861009(A1) 申请公布日期 2013.08.01
申请号 CA20132861009 申请日期 2013.01.25
申请人 INOTEK PHARMACEUTICALS CORPORATION 发明人 MCVICAR, WILLIAM K.
分类号 C07H19/167;A61K31/7076;A61P27/02;A61P27/06 主分类号 C07H19/167
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