发明名称 |
99mTc IMAGING AGENTS AND METHODS OF USE |
摘要 |
An embodiment of the invention comprises a ligand of Formula I wherein R1 and R2 are independently an alkyl or cycloalkyl; R3 is and alkyl; X is CO or SO2; Y is (CH2)n, C6H4, (OCH2CH2)n(NHCH2CH2)n and (OCH2CH2CH2)n, or a combination thereof; Z is linker group capable of conjugating to a vector; and n is an integer between 0 and 10. Also included are an imaging agent comprising a compound of Formula I complexed to 99mTc and their method of use to image a subject having a target site using single photon emission computed tomography (SPECT).
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申请公布号 |
US2013195756(A1) |
申请公布日期 |
2013.08.01 |
申请号 |
US201213362658 |
申请日期 |
2012.01.31 |
申请人 |
JOHNSON BRUCE FLETCHER;CARTER RANDALL LEE;RISHEL MICHAEL JAMES;DAREY MARK CHRISTOPHER PATRICK;WU TAO;YANG YANG;VALLIANT JOHN FITZMAURICE;STEPHENSON KARIN ANN;GENERAL ELECTRIC COMPANY |
发明人 |
JOHNSON BRUCE FLETCHER;CARTER RANDALL LEE;RISHEL MICHAEL JAMES;DAREY MARK CHRISTOPHER PATRICK;WU TAO;YANG YANG;VALLIANT JOHN FITZMAURICE;STEPHENSON KARIN ANN |
分类号 |
A61K51/04;A61K51/06;A61K51/08;A61K51/10;C07C235/84;C07C237/10;C07C311/18;C07C311/32;C07F13/00;C07K4/00;C07K14/00;C07K16/00 |
主分类号 |
A61K51/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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