发明名称 PROCESS FOR PREPARATION OF 3-[2-[4-(6-FLURO-1, 2-BENZISOXAZOL-3-YL)-1-PIPERIDTNYL]ETHYL]-6, 7, 8, 9-TETRAHYDRO-9-HYDROXY-2-METHYL-4H-PYRIODO[1, 2-A]PYRIMIDIN-4-ONE
摘要 A process for the preparation of paliperidone from the hydrolysis of paliperidone palmitate in the presence of an acid in a solvent.
申请公布号 WO2013080220(A3) 申请公布日期 2013.07.25
申请号 WO2012IN00771 申请日期 2012.11.26
申请人 DAVULURI, RAMMOHAN RAO 发明人 DAVULURI, RAMMOHAN RAO;PONNAIAH, RAVI;NEELA, PRAVEEN KUMAR;BATTHINI, GURUSWAMY;VENKATA NARASIMHARAO, TELEGAREDDY;RAVANABABU, KOSIREDDY;BANDLAMUDI, VEERANARAYANA
分类号 C07D471/04 主分类号 C07D471/04
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