发明名称 |
ACID ADDITION SALT OF A NORTRIPTYLINE-GABA CONJUGATE AND A PROCESS OF PREPARING SAME |
摘要 |
An acid addition salt of a nortriptyline-GABA conjugate, a novel crystalline form of a fumaric acid addition salt of a nortriptyline-GABA conjugate, and processes of preparing the forgoing are disclosed. Uses of the above-indicated forms of a nortriptyline-GABA conjugate in the treatment of CNS disorders, and in the treatment of pain in particular, are also disclosed. Further disclosed in a large-scale process of preparing a nortriptyline-GABA conjugate. |
申请公布号 |
US2013184347(A1) |
申请公布日期 |
2013.07.18 |
申请号 |
US201113825369 |
申请日期 |
2011.09.22 |
申请人 |
NUDELMAN ABRAHAM;REPHAELI ADA;GIL-AD IRIT;WEIZMAN ABRAHAM;SHAUL MAZAL;RAMOT AT TEL-AVIV UNIVERSITY LTD.;BIOLINERX LTD.;BAR-LLAN UNIVERSITY |
发明人 |
NUDELMAN ABRAHAM;REPHAELI ADA;GIL-AD IRIT;WEIZMAN ABRAHAM;SHAUL MAZAL |
分类号 |
C07C57/15;C07C51/41;C07C231/02;C07C231/12;C07C237/06 |
主分类号 |
C07C57/15 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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