发明名称 NOVEL HYDROXAMIC ACID DERIVATIVE
摘要 Provided is a novel compound which is useful as a pharmaceutical composition by inhibiting an LpxC activity, thereby exhibiting potent antimicrobial activity against gram-negative bacteria including Pseudomonas aeruginosa and its drug resistant bacteria. Provided is a hydroxamic acid derivative represented by the following general formula [1] or a pharmaceutically acceptable salt thereof:
申请公布号 KR20130079328(A) 申请公布日期 2013.07.10
申请号 KR20127025637 申请日期 2011.04.20
申请人 TAISHO PHARMACEUTICAL CO., LTD.;TOYAMA CHEMICAL CO., LTD. 发明人 TAKASHIMA HAJIME;TSURUTA RISA;YABUUCHI TETSUYA;OKA YUSUKE;URABE HIROKI;SUGA YOICHIRO;TAKAHASHI MASATO;UNEUCHI FUMITO;KOTSUBO HIRONORI;SHOJI MUNEO;KAWAGUCHI YASUKO
分类号 C07C235/56;A61K31/166;A61P31/04;C07D277/22 主分类号 C07C235/56
代理机构 代理人
主权项
地址