发明名称 |
B-DIHYDROFURAN DERIVING COMPOUND, METHOD FOR PRODUCING B-DIHYDROFURAN DERIVING COMPOUND OR B-TETRAHYDROFURAN DERIVING COMPOUND, B -GLYCOSIDE COMPOUND, METHOD FOR PRODUCING B-GLYCOSIDE COMPOUND, AND METHOD FOR PRODUCING 4'-ETHYNYL D4T AND ANALOGUE COMPOUNDS THEREOF |
摘要 |
The invention provides a process for producing a ²-dihydrofuran derivative represented by formula (1) or a ²-tetrahydrofuran derivative represented by formula (4), characterized in that the process includes causing a dialkyl dicarbonate, a diaralkyl dicarbonate, or a halide to act on a diol compound represented by formula (2) or (3). The invention also provides a process for producing 4'-ethynyl-2',3'-didehydro-3'-deoxythymidine or an analog thereof, the process including glycosylation and deprotection. |
申请公布号 |
EP2537839(A4) |
申请公布日期 |
2013.07.10 |
申请号 |
EP20110742187 |
申请日期 |
2011.02.07 |
申请人 |
NISSAN CHEMICAL INDUSTRIES, LTD. |
发明人 |
IRIYAMA, YUSUKE;HIGASHIYAMA, TSUTOMU |
分类号 |
C07D307/32;C07D405/04;C07H19/073 |
主分类号 |
C07D307/32 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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