发明名称 B-DIHYDROFURAN DERIVING COMPOUND, METHOD FOR PRODUCING B-DIHYDROFURAN DERIVING COMPOUND OR B-TETRAHYDROFURAN DERIVING COMPOUND, B -GLYCOSIDE COMPOUND, METHOD FOR PRODUCING B-GLYCOSIDE COMPOUND, AND METHOD FOR PRODUCING 4'-ETHYNYL D4T AND ANALOGUE COMPOUNDS THEREOF
摘要 The invention provides a process for producing a ²-dihydrofuran derivative represented by formula (1) or a ²-tetrahydrofuran derivative represented by formula (4), characterized in that the process includes causing a dialkyl dicarbonate, a diaralkyl dicarbonate, or a halide to act on a diol compound represented by formula (2) or (3). The invention also provides a process for producing 4'-ethynyl-2',3'-didehydro-3'-deoxythymidine or an analog thereof, the process including glycosylation and deprotection.
申请公布号 EP2537839(A4) 申请公布日期 2013.07.10
申请号 EP20110742187 申请日期 2011.02.07
申请人 NISSAN CHEMICAL INDUSTRIES, LTD. 发明人 IRIYAMA, YUSUKE;HIGASHIYAMA, TSUTOMU
分类号 C07D307/32;C07D405/04;C07H19/073 主分类号 C07D307/32
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