发明名称 PREPARATION OF EPTIFIBATIDE PEPTIDE
摘要 Provided is a process for the preparation of eptifibatide using a novel non-linear liquid phase peptide synthesis scheme. This invention makes use of combing precursor peptides synthesized separately in high purity and yield over presently known processes. The disclosed process has several advances over known processes like ease of scale-up and work-up as the process utilizes liquid phase peptide preparation chemistry.
申请公布号 WO2013057736(A3) 申请公布日期 2013.07.04
申请号 WO2012IN00386 申请日期 2012.06.04
申请人 EMCURE PHARMACEUTICALS LIMITED;GURJAR, MUKUND, KESHAV;PRAMANIK, CHINMOY;TRIPATHY, NARENDRA, KUMAR;ROY, ANUPAM, BADAL;CHAUDHARI, ASHOK, TUKARAM;BORHDE, AJIT, SAHEBRAO;KARHADE, GANESH, KALURAM;CHAGHULE, BALAJI, VASANT;MEHTA, SAMIT, SATISH;PAL, ARNAB ARUN 发明人 GURJAR, MUKUND, KESHAV;PRAMANIK, CHINMOY;TRIPATHY, NARENDRA, KUMAR;ROY, ANUPAM, BADAL;CHAUDHARI, ASHOK, TUKARAM;BORHDE, AJIT, SAHEBRAO;KARHADE, GANESH, KALURAM;CHAGHULE, BALAJI, VASANT;MEHTA, SAMIT, SATISH;PAL, ARNAB ARUN
分类号 C07K7/06;C07B57/00;C07C319/28;C07K1/02;C07K1/06;C07K5/09;C07K5/113 主分类号 C07K7/06
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