发明名称 |
PROCESS TO PREPARE ETHYL 4-METHYL-2-(4-(2-METHYLPROPYLOXY)-3-CYANOPHENYL)-5-THIAZOLECARBOXYLATE |
摘要 |
Disclosed is a process for the preparation of Ethyl 4-methyl-2-(4-(2-methylpropyloxy)-3-cyanophenyl)-5-thiazolecarboxylate (I) the key intermediate for the preparation of [2-[3-cyano-4-(2-Methyl-propoxy)phenyl]-4-methyl-5-thiazole carboxylic acid (Febuxostat, I(A)) is approved under the trademark Uloric® by the US Food and Drug Administration for the treatment of hyperuricemia and gouty arthritis.
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申请公布号 |
US2013172571(A1) |
申请公布日期 |
2013.07.04 |
申请号 |
US201013821094 |
申请日期 |
2010.09.08 |
申请人 |
KOMPELLA AMALA;GAMPA VENUE GOPALA KRISHNA;ADIBHATLA KALI SATYA BHUJANGA RAO;NANNAPANENI VENKAIAH CHOWDARY;NATCO PHARMA LIMITED |
发明人 |
KOMPELLA AMALA;GAMPA VENUE GOPALA KRISHNA;ADIBHATLA KALI SATYA BHUJANGA RAO;NANNAPANENI VENKAIAH CHOWDARY |
分类号 |
C07D277/56 |
主分类号 |
C07D277/56 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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