发明名称 NEW SALT AND MEDICAL USE
摘要 <P>PROBLEM TO BE SOLVED: To provide new treatments for gout that are more effective and/or are better tolerated. <P>SOLUTION: The invention provides 4-[2-(5-amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2- fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide or a pharmaceutically acceptable salt thereof for the treatment of a disease associated with elevated blood uric acid levels, such as hyperuricemia or gout. In another aspect the invention provides the tosylate salt of 4-[2-(5-amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide. <P>COPYRIGHT: (C)2013,JPO&INPIT
申请公布号 JP2013127010(A) 申请公布日期 2013.06.27
申请号 JP20130069382 申请日期 2013.03.28
申请人 PFIZER LTD 发明人 ALI ZAHID;BUTCHER KENNETH JOHN;BUTT RICHARD PHILIP;FELSTEAD STEPHEN JOHN;GLATT SOPHIE;MCKERNAN RUTH MITCHELL;PANESAR MANINDER
分类号 A61K31/427;A61K45/00;A61P19/06;A61P25/04;A61P29/00;A61P43/00;C07D417/12 主分类号 A61K31/427
代理机构 代理人
主权项
地址