发明名称 HYDROCHLORIDES AND HYDRATES OF 1-[(3-CYANOPYRIDIN-2-YL)METHYL]-3-METHYL-7-(2-BUTYN-1-YL)-8-(3-AMINOPIPERIDIN-1-YL)XANTHINE, THEIR PREPARATION AND THEIR USE AS MEDICAMENTS
摘要 <p>1-[(3-Cyano-pyridin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-(3-amino-piperidin-1-yl)-xanthine hydrochloride (I) is new. ACTIVITY : Neuroprotective; Nootropic; Cerebroprotective; Vasotropic; Antiarthritic; Antiarteriosclerotic; Anorectic; Antipsoriatic. MECHANISM OF ACTION : Dipeptidylpeptidase-IV inhibitor.</p>
申请公布号 EP1912990(B1) 申请公布日期 2013.06.26
申请号 EP20060777973 申请日期 2006.07.26
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH;BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG 发明人 PFRENGLE, WALDEMAR;SIEGER, PETER
分类号 C07D473/04;A61K31/522;A61P3/10 主分类号 C07D473/04
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