发明名称 |
HYDROCHLORIDES AND HYDRATES OF 1-[(3-CYANOPYRIDIN-2-YL)METHYL]-3-METHYL-7-(2-BUTYN-1-YL)-8-(3-AMINOPIPERIDIN-1-YL)XANTHINE, THEIR PREPARATION AND THEIR USE AS MEDICAMENTS |
摘要 |
<p>1-[(3-Cyano-pyridin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-(3-amino-piperidin-1-yl)-xanthine hydrochloride (I) is new. ACTIVITY : Neuroprotective; Nootropic; Cerebroprotective; Vasotropic; Antiarthritic; Antiarteriosclerotic; Anorectic; Antipsoriatic. MECHANISM OF ACTION : Dipeptidylpeptidase-IV inhibitor.</p> |
申请公布号 |
EP1912990(B1) |
申请公布日期 |
2013.06.26 |
申请号 |
EP20060777973 |
申请日期 |
2006.07.26 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH;BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG |
发明人 |
PFRENGLE, WALDEMAR;SIEGER, PETER |
分类号 |
C07D473/04;A61K31/522;A61P3/10 |
主分类号 |
C07D473/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|