发明名称 |
PROCESS FOR THE PREPARATION OF (1R,4R)-6'-FLUORO-(N,N-DIMETHYL- AND N-METHYL)-4-PHENYL-4',9'-DIHYDRO-3'H-SPIRO[CYCLOHEXANE-1,1'-PYRANO-[3,4,B]INDOL]-4-AMINE |
摘要 |
<p>The present invention relates to a process for the preparation of (1r,4r)-6'-fluoro-N,N-dimethyl-4-phenyl-4',9'-dihydro-3'H-spiro[cyclohexane-1,1'-pyrano[3,4b]indol]-4-amine and (1r,4r)-6'-fluoro-N-methyl-4-phenyl-4',9'-dihydro-3'H-spiro[cyclohexane-1,1'-pyrano[3,4b]- indol]-4-amine or physiologically acceptable acid addition salts thereof.</p> |
申请公布号 |
WO2013087589(A1) |
申请公布日期 |
2013.06.20 |
申请号 |
WO2012EP75002 |
申请日期 |
2012.12.11 |
申请人 |
GRUENENTHAL GMBH |
发明人 |
PRUEHS, STEFAN;GRIEBEL, CARSTEN;HELL, WOLFGANG |
分类号 |
C07D491/107 |
主分类号 |
C07D491/107 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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