发明名称 PROCESS FOR THE PREPARATION OF (5-FLUORO-2-METHYL-3-QUINOLIN-2-YLMETHYL-INDOL-1-YL)-ACETIC ACID ESTERS
摘要 <p>The invention relates to a process for the preparation of a compound of formula (I) wherein R1 is C1C6 alkyl or benzyl by reacting a compound of formula (II) wherein R1 is as defined for formula (I) with 2-quinoline carboxaldehyde. The process is suitable for use on an industrial scale.</p>
申请公布号 WO2013088108(A1) 申请公布日期 2013.06.20
申请号 WO2012GB00903 申请日期 2012.12.14
申请人 OXAGEN LIMITED 发明人 TONNEL, JACQUES;PINTUS, TONY;BURGOS, ALAIN
分类号 C07D401/06 主分类号 C07D401/06
代理机构 代理人
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