发明名称 |
PROCESS FOR THE PREPARATION OF (5-FLUORO-2-METHYL-3-QUINOLIN-2-YLMETHYL-INDOL-1-YL)-ACETIC ACID ESTERS |
摘要 |
<p>The invention relates to a process for the preparation of a compound of formula (I) wherein R1 is C1C6 alkyl or benzyl by reacting a compound of formula (II) wherein R1 is as defined for formula (I) with 2-quinoline carboxaldehyde. The process is suitable for use on an industrial scale.</p> |
申请公布号 |
WO2013088108(A1) |
申请公布日期 |
2013.06.20 |
申请号 |
WO2012GB00903 |
申请日期 |
2012.12.14 |
申请人 |
OXAGEN LIMITED |
发明人 |
TONNEL, JACQUES;PINTUS, TONY;BURGOS, ALAIN |
分类号 |
C07D401/06 |
主分类号 |
C07D401/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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