发明名称 PROCESS FOR THE PREPARATION OF ENANTIOMERIC FORMS OF 2,3-DIAMINOPROPIONIC ACID DERIVATIVES
摘要 <p>The disclosure relates to a process for the preparation of the enantiomeric forms of 2,3-diaminopropionic acid derivatives of formula I, wherein R1, R2 and R3 are defined as in the disclosure, by racemate resolution. The separation of the racemate into its enantiomers takes place through formation of diastereomeric salts upon addition of an enantiomerically pure auxiliary, and subsequent separation by fractional crystallization.</p>
申请公布号 EP2603491(A1) 申请公布日期 2013.06.19
申请号 EP20110743050 申请日期 2011.08.05
申请人 SANOFI 发明人 GRAF, CLAUS-DIETER;RIEKE-ZAPP, JOERG
分类号 C07D213/74;C07D239/42 主分类号 C07D213/74
代理机构 代理人
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