发明名称 |
Chemical linkers and cleavable substrates and conjugates thereof |
摘要 |
The present disclosure provides drug-ligand conjugates and drug-cleavable substrate conjugates that are potent cytotoxins. The disclosure is also directed to compositions containing the drug-ligand conjugates, and to methods of treatment using them.
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申请公布号 |
US8461117(B2) |
申请公布日期 |
2013.06.11 |
申请号 |
US20070521391 |
申请日期 |
2007.12.28 |
申请人 |
SUFI BILAL;GUERLAVAIS VINCENT;CHEN LIANG;GANGWAR SANJEEV;ZHANG QIAN;PASSMORE DAVID B.;MEDAREX, INC. |
发明人 |
SUFI BILAL;GUERLAVAIS VINCENT;CHEN LIANG;GANGWAR SANJEEV;ZHANG QIAN;PASSMORE DAVID B. |
分类号 |
A61K38/00;A61K38/10;A61P35/00;A61P35/02;A61P35/04 |
主分类号 |
A61K38/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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