发明名称 |
AGENT FOR ANTIPLATELET, ANTI-INFLAMMATORY AND CYTOPROTECTIVE THERAPY |
摘要 |
FIELD: medicine, pharmaceutics.SUBSTANCE: invention refers to medicine, and concerns an agent for prevention and treatment of cardiovascular diseases. The peptide 3-mercaptopropionyl-Phe-Ile-lle-Arg-Lys-Pro-Asp-Lys-NHis synthetised which has greater availability and lower price than known analogues; it possesses the antiplatelet, anti-inflammatory and cytoprotective properties.EFFECT: invention provides reduced spontaneous thrombocyte aggregation, inflammation inhibition by reducing histamine secretion, cell protection against neurotoxic actions of thrombin.1 cl, 4 ex |
申请公布号 |
RU2483746(C1) |
申请公布日期 |
2013.06.10 |
申请号 |
RU20120120386 |
申请日期 |
2012.05.17 |
申请人 |
FEDERAL'NOE GOSUDARSTVENNOE UNITARNOE PREDPRIJATIE "GOSUDARSTVENNYJ NAUCHNYJ TSENTR "NAUCHNO-ISSLEDOVATEL'SKIJ INSTITUT ORGANICHESKIKH POLUPRODUKTOV I KRASITELEJ" (FGUP "GNTS "NIOPIK") |
发明人 |
RUMSH LEV DAVYDOVICH;STRUKOVA SVETLANA MIKHAJLOVNA;GORBACHEVA LJUBOV' RUFEHL'EVNA;BESPALOVA ZHANNA DMITRIEVNA;SIDOROVA MARIJA VLADIMIROVNA;FRID DMITRIJ ALEKSANDROVICH;FEL'DMAN BORIS MORDKOVICH;BURJACHKOVSKAJA LJUDMILA IVANOVNA |
分类号 |
A61K38/00;A61K38/46;A61P29/00 |
主分类号 |
A61K38/00 |
代理机构 |
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代理人 |
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地址 |
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