发明名称 |
PYRIDINE AND PYRIMIDINE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE |
摘要 |
This invention comprises the novel compounds of formula (I) wherein R1, R2, R3 and X have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
|
申请公布号 |
US2013143898(A1) |
申请公布日期 |
2013.06.06 |
申请号 |
US201213347338 |
申请日期 |
2012.01.10 |
申请人 |
BERNADETTE MARCONNET-DECRANE LAURENCE FRANCOISE;DOMINIQUE GAURRAND SANDRINE FRANCOISE;ANGIBAUD PATRICK RENE;JANSSEN PHARMACEUTICA N.V. |
发明人 |
BERNADETTE MARCONNET-DECRANE LAURENCE FRANCOISE;DOMINIQUE GAURRAND SANDRINE FRANCOISE;ANGIBAUD PATRICK RENE |
分类号 |
C07D213/82;A61K31/496;A61K45/06 |
主分类号 |
C07D213/82 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|