摘要 |
C:/NRPortbl/DCC/ALHm2932546_m..juuL - 4IU/zU I U The present invention provides compounds having formula (I), and additionally provides methods for the synthesis thereof and methods for the use thereof in the treatment of various disorders including inflammatory or autoimmune disorders, and disorders involving malignancy or increased angiogenesis, wherein RI-RI1 , t, X, Y, Z, and n are as defined herein. R10 O R3 JR2 n ORS n R7 Re |
申请人 |
EISAI R&D MANAGEMENT CO., LTD. |
发明人 |
HARMANGE, JEAN-CHRISTOPHE;SHIROTA, HIROSHI;TANAKA, ISAO;MURAMOTO, KENZO;KUBOI, YOSHIKAZU;DU, HONG;LEMELIN, CHARLES-ANDRE;SHEN, YONG-CHUN;KIMURA, AKIFUMI;BOIVIN, ROCH;SPYVEE, MARK;KAWADA, MEGUMI;WANG, JOHN (YUAN);FUJITA, MASANORI;GUSOVSKY, FABIAN;KAWAI, TAKATOSHI;SUKURAI, HIDEKI;EGUCHI, YOSHIHITO;GOTO, MASAKI;KAWAKAMI, YOSHIYUKI;MIZUI, YOSHIHARU;YAMAMOTO, SATOSHI;JIANG, YIMIN;MATSUSHIMA, TOMOHIRO;LI, XIANG-YI;YONEDA, NAOKI;CHOW, JESSE;INOUE, ATSUSHI;KOTAKE, MAKOTO;CHIBA, KENICHI |