发明名称 DUAL NK1/NK3 ANTAGONIST AGAINST SCHIZOPHRENIA
摘要 THE PRESENT INVENTION RELATES TO THE USE OF COMPOUNDS OF THE GENERAL FORMULA ?: WHEREIN R� IS LOWER ALKYL OR HALOGEN; R� IS HYDROGEN OR HALOGEN;R� -(CHR')nOH, PHENYL, OPTIONALLY SUBSTITUTED BY -(CHR')nOH, OR IS A SATURATED, PARTIAL SATURATED OR AROMATIC 5-OR 6-MEMBERED HETEROCYCLIC RING WITH ONE HETEROATOM, SELECTED FROM THE GROUP CONSISTING OF-N(R?)-,-N=,_N_=, -S- OR -S(O)?, AND WHICH RINGS ARE OPTIONALLY SUBSTITUTED BY?(CHR')nOH; R' IS INDEPENDENTLY FROM "n" HYDROGEN OR -(CH?)nOH; R? IS HYDROGEN, -S(O?)-LOWER ALKYL OR -C(O)-LOWER ALKYL; X IS ?O-, -CH?O-, -S- OR A BOND; n IS 1 OR 2; OR TO PHARMACEUTICALLY ACTIVE ACID-ADDITION SALTS THEREOF, FOR THE PREPARATION OF MEDICAMENTS FOR THE TREATMENT OF SCHIZOPHRENIA.
申请公布号 MY148684(A) 申请公布日期 2013.05.31
申请号 MY2005PI03652 申请日期 2005.08.05
申请人 F. HOFFMANN-LA ROCHE AG 发明人 PATRICK SCHNIDER
分类号 A61K31/44;A61K31/4436;A61K31/4439;A61K31/444;A61P25/18;C07D213/82 主分类号 A61K31/44
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