发明名称 |
Novel naphthyridine derivative monohydrate and method for producing the same |
摘要 |
Disclosed is 1-(2-(4-((2,3-dihydro(1,4)dioxino(2,3-c)pyridin-7-ylmethyl)amino)piperidin-1-yl)ethyl)-7-fluoro-1,5-naphthyridin-2(1H)-one monohydrate, which has a strong antibacterial activity. The compound is highly safe and useful as an original drug for pharmaceutical preparations. Also disclosed is a method which is useful for producing 1-(2-(4-((2,3-dihydro(1,4)dioxino(2,3-c)pyridin-7-ylmethyl)amino)piperidin-1-yl)ethyl)-7-fluoro-1,5-naphthyridin-2(1H)-one monohydrate. |
申请公布号 |
AU2008330725(B2) |
申请公布日期 |
2013.05.30 |
申请号 |
AU20080330725 |
申请日期 |
2008.11.25 |
申请人 |
TAISHO PHARMACEUTICAL CO., LTD.;TOYAMA CHEMICAL CO., LTD. |
发明人 |
KIYOTO, TARO;HORIKIRI, HIROMASA;BABA, YASUTAKA;USHIYAMA, FUMIHITO;SYOJI, MUNEO;TAKEBAYASHI, MASAHIRO;URABE, HIROKI;NOGUCHI, TOSHIYA |
分类号 |
C07D519/00;A61K31/4545;A61P31/04;C07D309/40;C07D491/056 |
主分类号 |
C07D519/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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