发明名称 HETEROARYL-PYRAZOLE DERIVATIVE
摘要 A compound represented by formula [I] and a pharmaceutically accepted salt of said compound are a novel compound and a pharmaceutically accepted salt thereof which exert antagonistic activity against group II metabotropic glutamate (mGlu) receptors, and are effective as a novel preventive or therapeutic agent for disorders such as mood disorders (depressive disorder, bipolar disorder, etc.), anxiety disorders (generalized anxiety disorder, panic disorder, obsessive-compulsive disorder, social anxiety disorder, posttraumatic stress disorder, a specific phobic disorder, acute stress disorder, etc.), schizophrenia, Alzheimer's disease, cognitive impairment, dementia, drug dependence, convulsions, shivering, pain, sleep disorders, and the like.
申请公布号 US2013137865(A1) 申请公布日期 2013.05.30
申请号 US201113814869 申请日期 2011.08.11
申请人 NAKAMURA TOSHIO;SAKAGAMI KAZUNARI;KONISHI KAZUHIDE;YAMAMOTO KANAKO;MASUDA SEIJI;MATSUDA YOHEI;OKADA KUMIKO;SHIBATA TSUYOSHI;OHTA HIROSHI;YASUHARA AKITO;KAWAMOTO HIROSHI;AMADA HIDEAKI;URABE HIROKI;NISHIKAWA RIE;KASHIWA ASHIWA SHUHEI;TAISHO PHARMACEUTICAL CO., LTD. 发明人 NAKAMURA TOSHIO;SAKAGAMI KAZUNARI;KONISHI KAZUHIDE;YAMAMOTO KANAKO;MASUDA SEIJI;MATSUDA YOHEI;OKADA KUMIKO;SHIBATA TSUYOSHI;OHTA HIROSHI;YASUHARA AKITO;KAWAMOTO HIROSHI;AMADA HIDEAKI;URABE HIROKI;NISHIKAWA RIE;KASHIWA ASHIWA SHUHEI
分类号 C07D413/14;C07D231/38;C07D403/04;C07D413/04 主分类号 C07D413/14
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