发明名称 |
7-substituted indole MCL-1 inhibitors |
摘要 |
Compounds which inhibit the activity of anti-apoptotic Mcl-1 protein, compositions containing the compounds, and methods of treating diseases involving overexpressed or unregulated Mcl-1 protein are disclosed.
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申请公布号 |
US8445679(B2) |
申请公布日期 |
2013.05.21 |
申请号 |
US20080104294 |
申请日期 |
2008.04.16 |
申请人 |
WANG XILU;SONG XIAOHONG;ELMORE STEVEN W.;BRUNCKO MILAN;MADAR DAVID J.;SOUERS ANDREW J.;HASVOLD LISA A.;WANG LE;TAO ZHI-FU;KUNZER AARON K.;ABBVIE INC. |
发明人 |
WANG XILU;SONG XIAOHONG;ELMORE STEVEN W.;BRUNCKO MILAN;MADAR DAVID J.;SOUERS ANDREW J.;HASVOLD LISA A.;WANG LE;TAO ZHI-FU;KUNZER AARON K. |
分类号 |
C07D403/04;A61K31/497 |
主分类号 |
C07D403/04 |
代理机构 |
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代理人 |
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地址 |
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