发明名称 N, N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS
摘要 THE PRESENT INVENTION PROVIDES A PYRROLIDINE COMPOUND OF GENERAL FORMULA (1) OR A SALT THEREOF, WHEREIN R¹º¹ AND R¹º² ARE EACH INDEPENDENTLY A PHENYL GROUP OR A PYRIDYL GROUP, THE PHENYL GROUP OR THE PYRIDYL GROUP MAY HAVE ONE OR MORE SUBSTITUENTS SELECTED FROM HALOGEN ATOMS AND LOWER ALKYL GROUPS OPTIONALLY SUBSTITUTED WITH ONE OR MORE HALOGEN ATOMS, ETC. THE PYRROLIDINE COMPOUND OR A SALT THEREOF OF THE PRESENT INVENTION IS USABLE TO PRODUCE A PHARMACEUTICAL PREPARATION HAVING A WIDER THERAPEUTIC SPECTRUM AND BEING CAPABLE OF EXHIBITING SUFFICIENT THERAPEUTIC EFFECTS AFTER SHORT-TERM ADMINISTRATION.
申请公布号 MY148653(A) 申请公布日期 2013.05.15
申请号 MY2006PI02198 申请日期 2006.05.11
申请人 OTSUKA PHARMACEUTICAL CO., LTD. 发明人 MUNEAKI KURIMURA;YOHJI SAKURAI;AKIHITO WATANABE;YASUYO SAKATA;TAKUMI MASUMOTO;KOHEI AKAZAWA;HARUHIKO SUGINO;NAOKI AMADA;SATOSHI OHASHI;TOMOICHI SHINOHARA;HIROFUMI SASAKI;SHINICHI TAIRA;CHISAKO MORITA;JUNKO YAMASHITA;SATOKO NAKAJIMA;TAKAHIRO TOMOYASU;NOBUAKI ITO;KUNINORI TAI;NORIAKI TAKEMURA;TAKAYUKI MATSUZAKI;YASUHIRO MENJO;SHIN MIYAMURA
分类号 A61K31/40 主分类号 A61K31/40
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