发明名称 MODULATORS OF LXR
摘要 Compounds, compositions and methods for modulating the activity of nuclear receptors are provided. In particular, heterocyclic compounds are provided for modulating the activity of nuclear receptors, including liver X receptor (LXR) and orphan nuclear receptors. In certain embodiments, the compounds are N-substituted pyridones.
申请公布号 EP1465869(B1) 申请公布日期 2013.05.15
申请号 EP20020787071 申请日期 2002.12.20
申请人 EXELIXIS PATENT COMPANY LLC 发明人 BAYNE, CHRISTOPHER, D.;JOHNSON, ALAN, T.;LU, SHAO-PO;MOHAN, RAJU;GRIFFITH, RONALD, C.
分类号 C07D213/64;A61K31/437;A61K31/4375;A61K31/4412;A61K31/4418;A61K31/443;A61K31/4433;A61K31/4436;A61K31/4439;A61K31/4545;A61K31/496;A61K31/497;A61P1/16;A61P3/04;A61P3/06;A61P3/10;A61P7/00;A61P9/10;A61P17/02;A61P25/16;A61P25/28;A61P29/00;A61P35/00;A61P43/00;C07D213/80;C07D213/84;C07D213/85;C07D213/89;C07D401/04;C07D401/06;C07D401/12;C07D405/04;C07D405/06;C07D405/10;C07D405/12;C07D409/04;C07D413/06;C07D417/04;C07D417/06;C07D417/12;C07D471/04 主分类号 C07D213/64
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