发明名称 Heteroaryls and uses thereof
摘要 This invention provides compounds of formula I: wherein R1, R2, CY, Y1, Y2, X1, X2, and X3 are as described in the specification. The compounds are inhibitors of PI3K and are thus useful for treating proliferative, inflammatory, or cardiovascular disorders.
申请公布号 US8440664(B2) 申请公布日期 2013.05.14
申请号 US201213449341 申请日期 2012.04.18
申请人 CARDIN DAVID P.;GAULIN JEFFREY;GREENSPAN PAUL;RENOU CHRISTELLE C.;VYSKOCIL STEPAN;XU TIANLIN;MILLENNIUM PHARMACEUTICALS, INC. 发明人 CARDIN DAVID P.;GAULIN JEFFREY;GREENSPAN PAUL;RENOU CHRISTELLE C.;VYSKOCIL STEPAN;XU TIANLIN
分类号 A61K31/535 主分类号 A61K31/535
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