发明名称 AZOLE DERIVATIVE
摘要 The invention according to the present application provides a therapeutic or prophylactic agent for diseases including mood disorders, anxiety disorders, schizophrenia, Alzheimer's disease, Parkinson's disease, Huntington's chorea, eating disorder, hypertension, digestive diseases, drug dependence, epilepsy, cerebral infarction, cerebral ischemia, cerebral edema, head injury, inflammations, immune-related diseases and alopecia. Specifically provided is an azole derivative having an arginine-vasopressin 1b receptor antagonistic activity and represented by general formula (I) or a pharmaceutically acceptable salt thereof.
申请公布号 WO2013062027(A1) 申请公布日期 2013.05.02
申请号 WO2012JP77541 申请日期 2012.10.25
申请人 TAISHO PHARMACEUTICAL CO., LTD. 发明人 YOSHINAGA, MITSUKANE;KUWADA, TAKESHI;MIYAKOSHI, NAOKI;ISHIZAKA, TOMOKO;WAKASUGI, DAISUKE;SHIROKAWA, SHIN-ICHI;HATTORI, NOBUTAKA;SHIMAZAKI, YOUICHI
分类号 C07D207/444;A61K31/4164;A61K31/4178;A61K31/4196;A61K31/4439;A61K31/444;A61K31/454;A61K31/4545;A61K31/46;A61K31/4725;A61K31/496;A61K31/537;A61K31/5377;A61K31/5386;A61K31/541;A61K31/553;A61P1/04;A61P9/10;A61P9/12;A61P17/14;A61P25/00;A61P25/08;A61P25/14;A61P25/16;A61P25/18;A61P25/22;A61P25/28;A61P25/30;A61P29/00;A61P37/02;A61P43/00;C07D231/12;C07D233/64;C07D233/70;C07D249/08;C07D249/10;C07D263/32;C07D277/20;C07D277/30;C07D401/04;C07D401/10;C07D403/04;C07D403/06;C07D403/10;C07D413/10;C07D451/06;C07D491/107;C07D498/08 主分类号 C07D207/444
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