发明名称 Crystalline form of eszopiclone, composition, preparation and uses thereof
摘要 The present invention discloses a crystalline form of S-zopiclone (Formula I) having a powder X-Ray diffraction spectrum excited by Cu-Ka radiation with characteristic peaks expressed in terms of 2theta at about 11.08°, about 12.38°, about 15.86°, about 17.88°, about 19. 98° and about 20.58°; a DSC thermogram with a peak at about 207.7° C. and an infrared absorption spectrum (IR) with characteristic peaks at about 3078 cm-1, about 2942~2838 cm-1, about 2790 cm-1, about 1716 cm-1, about 1463 cm-1, about 1372 cm-1 and about 757 cm-1. The present invention also discloses a method for preparing the crystalline form of eszopiclone, its pharmaceutical composition and its use in preparing a medicament for treating sleep disorders.
申请公布号 US8431577(B2) 申请公布日期 2013.04.30
申请号 US20090999867 申请日期 2009.04.17
申请人 WANG GUOCHENG;XU XUEYU;TIANJIN TASLY GROUP CO., LTD. 发明人 WANG GUOCHENG;XU XUEYU
分类号 A61K31/495 主分类号 A61K31/495
代理机构 代理人
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