发明名称 |
SUBSTITUTED OXADIAZOLYL PYRIDINONES AND OXADIAZOLYL PYRIDAZINONES AS HIF INHIBITORS |
摘要 |
The present application relates to novel substituted 5-(1,2,4-oxadiazolo-5-yl) pyridine-2-ones and 6-(1,2,4-oxadiazolo-5-yl) pyridazine-3-ones, a method for preparation thereof, the use thereof for treatment and/or prevention of diseases, and for producing medicines for the treatment and/or prevention of diseases, in particular for treating and/or preventing hyperproliferative and angiogenic disorders, and disorders that are caused by a metabolic adaptation to hypoxic conditions. Such treatments can be carried out as monotherapy or in combination with other medicines or additional therapeutic measures. |
申请公布号 |
WO2013057101(A1) |
申请公布日期 |
2013.04.25 |
申请号 |
WO2012EP70484 |
申请日期 |
2012.10.16 |
申请人 |
BAYER INTELLECTUAL PROPERTY GMBH |
发明人 |
HAERTER, MICHAEL;BECK, HARTMUT;ELLINGHAUS, PETER;UNTERSCHEMMANN, KERSTIN |
分类号 |
C07D413/04;A61K31/4245;C07D413/14 |
主分类号 |
C07D413/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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