发明名称 Arylethynyl derivatives
摘要 The present invention relates to ethynyl compounds of formula I wherein R1, R2, R2′, R3, R3′, R4, R4′, U, V, W, Y, m, and n are as defined herein and to a pharmaceutically acceptable acid addition salts, to a racemic mixtures, or to its corresponding enantiomers and/or optical isomers and/or stereoisomers thereof. Compounds of formula I are allosteric modulators of the metabotropic glutamate receptor subtype 5 (mGluR5).
申请公布号 US8420661(B2) 申请公布日期 2013.04.16
申请号 US201113066044 申请日期 2011.04.05
申请人 GREEN LUKE;GUBA WOLFGANG;JAESCHKE GEORG;JOLIDON SYNESE;LINDEMANN LOTHAR;RICCI ANTONIO;RUEHER DANIEL;STADLER HEINZ;VIEIRA ERIC;HOFFMANN-LA ROCHE INC. 发明人 GREEN LUKE;GUBA WOLFGANG;JAESCHKE GEORG;JOLIDON SYNESE;LINDEMANN LOTHAR;RICCI ANTONIO;RUEHER DANIEL;STADLER HEINZ;VIEIRA ERIC
分类号 C07D211/00;A61K31/44;A61K31/70;C07D211/68;C07D211/80;C07D213/00;C07D213/02;C07D215/00;C07D217/00;C07D219/00;C07D221/00;C07D401/00;C07D405/00;C07D409/00;C07D411/00;C07D413/00;C07D417/00;C07D419/00;C07D421/00 主分类号 C07D211/00
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