发明名称 SUBSTITUTED 6-CYCLOHEXYLALKYL SUBSTITUTED 2-QUINOLINONES AND 2-QUINOXALINONES AS POLY(ADP-RIBOSE) POLYMERASE INHIBITORS
摘要 <p num="1"><br/><br/><br/>The present invention provides compounds of formula (I), their use as PARP <br/>inhibitors as well as pharmaceutical compositions comprising said compounds of <br/>formula (I) wherein n, s, R1, R2, R3, Q, X and Y have defined meanings.<br/>
申请公布号 CA2548273(C) 申请公布日期 2013.04.16
申请号 CA20042548273 申请日期 2004.11.18
申请人 JANSSEN PHARMACEUTICA N.V. 发明人 MABIRE, DOMINIQUE JEAN-PIERRE;VAN DUN, JACOBUS ALPHONSUS JOSEPHUS;SOMERS, MARIA VICTORINA FRANCISCA;WOUTERS, WALTER BOUDEWIJN LEOPOLD
分类号 C07D241/44;A61K31/498;A61P43/00;C07D215/22;C07D215/227;C07D401/06;C07D401/14;C07D409/14;C07D491/10 主分类号 C07D241/44
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