发明名称 |
SUBSTITUTED 6-CYCLOHEXYLALKYL SUBSTITUTED 2-QUINOLINONES AND 2-QUINOXALINONES AS POLY(ADP-RIBOSE) POLYMERASE INHIBITORS |
摘要 |
<p num="1"><br/><br/><br/>The present invention provides compounds of formula (I), their use as PARP <br/>inhibitors as well as pharmaceutical compositions comprising said compounds of <br/>formula (I) wherein n, s, R1, R2, R3, Q, X and Y have defined meanings.<br/>
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申请公布号 |
CA2548273(C) |
申请公布日期 |
2013.04.16 |
申请号 |
CA20042548273 |
申请日期 |
2004.11.18 |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
MABIRE, DOMINIQUE JEAN-PIERRE;VAN DUN, JACOBUS ALPHONSUS JOSEPHUS;SOMERS, MARIA VICTORINA FRANCISCA;WOUTERS, WALTER BOUDEWIJN LEOPOLD |
分类号 |
C07D241/44;A61K31/498;A61P43/00;C07D215/22;C07D215/227;C07D401/06;C07D401/14;C07D409/14;C07D491/10 |
主分类号 |
C07D241/44 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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