发明名称 |
SOLID-PHASE FLUORINATION OF BENZOTHIAZOLES |
摘要 |
The invention provides a process for the production of an 18F-labelled tracer which comprises treatment of a solid support-bound precursor of formula (I) SOLID SUPPORT-LINKER-X-TRACER  (I) wherein X is a group which promotes nucleophilic substitution at a specific site on the attached TRACER and the TRACER is of formula (A) |
申请公布号 |
US2013089501(A1) |
申请公布日期 |
2013.04.11 |
申请号 |
US201213687485 |
申请日期 |
2012.11.28 |
申请人 |
GE HEALTHCARE LIMITED;HAMMERSMITH IMANET LIMITED;HAMMERSMITH IMANET LIMITED;GE HEALTHCARE LIMITED |
发明人 |
BRADY FRANK;LUTHRA SAJINDER KAUR;GIBSON ALEXANDER MARK |
分类号 |
C07B59/00;A61K51/04;C07D277/66 |
主分类号 |
C07B59/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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