发明名称 METHOD FOR PREPARING INTERMEDIATE OF SITAGLIPTIN USING CHIRAL OXIRANE
摘要 Disclosed is: a novel, simple and low-cost method for preparing 3-hydroxy-4-(2,4,5-trifluorophenyl)-butyric acid, particularly (3S)-3-hydroxy-4-(2,4,5-trifluorophenyl)-butyric acid, which is used as a key intermediate in the preparation of sitagliptin.
申请公布号 KR101253106(B1) 申请公布日期 2013.04.10
申请号 KR20090093894 申请日期 2009.10.01
申请人 发明人
分类号 C07C51/08;C07C59/56;C07C255/36;C07D303/08 主分类号 C07C51/08
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