发明名称 Use of cyclic depsipeptides to inhibit kallikrein 7
摘要 The present application relates to cyclic depsipeptides of Formula I: or derivatives thereof, wherein X, A1, A2, A3, A4, A5, A6 and A7 are defined herein. The cyclic depsipeptides of Formula I are inhibitors of kallikrein 7 and thus can be employed for the treatment of kallikrein-7 dependent diseases.
申请公布号 US8415305(B2) 申请公布日期 2013.04.09
申请号 US20080673785 申请日期 2008.08.14
申请人 KRASTEL PHILIPP;LIECHTY BRIGITTA-MARIA;SCHMITT ESTHER;SCHREINER ERWIN PAUL;NOVARTIS AG 发明人 KRASTEL PHILIPP;LIECHTY BRIGITTA-MARIA;SCHMITT ESTHER;SCHREINER ERWIN PAUL
分类号 A61K38/12;A61P17/00;A61P17/04;A61P17/06;C07K7/54 主分类号 A61K38/12
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