发明名称 |
5 - BENZYLAMINOMETHYL - 6 - AMINOPYRAZOLO [3, 4 -B] PYRIDINE DERIVATIVES AS CHOLESTERYL ESTER -TRANSFER PROTEIN (CETP) INHIBITORS USEFUL FOR THE TREATMENT OF ATHEROSCLEROSIS |
摘要 |
The present application relates to a series of substituted pyra- zolopyridin-6-amines having the general formula (I), including their stereoisomers and/or their pharmaceutically acceptable salts. Wherein R, R1, R2, Ra, Raa, Rb and n are as defined herein. The present invention further relates to pharmaceutical compositions comprising compounds of formula (I). The compounds of this application are useful as CETP inhibitors for increasing HDL cholesterol and decreasing LDL cholesterol in a patient. |
申请公布号 |
WO2013046045(A1) |
申请公布日期 |
2013.04.04 |
申请号 |
WO2012IB02435 |
申请日期 |
2012.09.27 |
申请人 |
DR. REDDY'S LABORATORIES, LTD. |
发明人 |
BORUAH, ANIMA;ALIKUNJU, SHANAVAS |
分类号 |
C07D471/04;A61K31/437;A61K31/444;A61K31/506;A61P9/10 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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