发明名称 PYRAZOLE DERIVATIVES USED AS CCR4 RECEPTOR ANTAGONISTS
摘要 Disclosed is a compound of formula (I) or a salt thereof such as N-[(3-{ [3-{ [(5-Chloro-2-thienyl)sulfonyl]amino} -4-(methyloxy)-1H-indazol-1-yl]methyl} phenyl)methyl]-2-hydroxy-2-methylpropanamide, which is useful for treating a disease associated with CCR4 receptor antagonist. Also disclosed is the process of the preparation of compound formula (I).
申请公布号 NZ594641(A) 申请公布日期 2013.03.28
申请号 NZ20100594641 申请日期 2010.02.24
申请人 GLAXO GROUP LIMITED 发明人 HOBBS, HEATHER;HODGSON, SIMON, TEANBY;LACROIX, YANNICK, MAURICE;NEEDHAM, DEBORAH;PARR, NIGEL, JAMES;PROCOPIOU, PANAYIOTIS, ALEXANDROU;RITCHIE, TIMOTHY, JOHN;WOODROW, MICHAEL, DAVID
分类号 C07D231/56;A61K31/381;A61K31/416;A61P11/06;A61P11/08;A61P29/00;A61P37/08;C07D409/12;C07D409/14 主分类号 C07D231/56
代理机构 代理人
主权项
地址