发明名称 METHOD FOR PREPARING Beta-ARTEMETHER
摘要 <p>Provided is a method for synthesizing beta-Artemether. The method uses dihydroartemisinin as a raw material, which has an etherifying reaction with trimethyl orthoformate in an organic solvent in the presence of catalyst, to give beta-Artemether, with a byproduct alpha-Artemether content of less than 6%.</p>
申请公布号 WO2013040750(A1) 申请公布日期 2013.03.28
申请号 WO2011CN79858 申请日期 2011.09.20
申请人 SHANGHAI DESANO PHARMACEUTICALS INVESTMENT CO., LTD;SHANGHAI DESANO CHEMICAL PHARMACEUTICAL CO., LTD.;JIANGSU PUXIN PHARMACEUTICALS DEVELOPMENT CO., LTD;LI, JINLIANG;ZHAO, NAN;JIANG, FEI;ZHENG, YUQING;YAO, XIAOGUANG 发明人 LI, JINLIANG;ZHAO, NAN;JIANG, FEI;ZHENG, YUQING;YAO, XIAOGUANG
分类号 C07D493/18;A61P33/06 主分类号 C07D493/18
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