The presently disclosed subject matter provides methods of preparing synthetic prostacyclin analogues, including Beraprost, either as racemic mixtures or as single stereoisomers. Also provided are novel synthetic intermediates for use in these methods.
申请公布号
WO2013040068(A2)
申请公布日期
2013.03.21
申请号
WO2012US54910
申请日期
2012.09.12
申请人
IRIX PHARMACEUTICALS, INC.;YIANNIKOUROS, GEORGE PETROS;KALARITIS, PANOS;GAMAGE, CHAMINDA PRIYAPUSHPA;AREFYEV, DENIS VIKTOROVICH
发明人
YIANNIKOUROS, GEORGE PETROS;KALARITIS, PANOS;GAMAGE, CHAMINDA PRIYAPUSHPA;AREFYEV, DENIS VIKTOROVICH