发明名称 BENZONITRILE DERIVATIVES AS KINASE INHIBITORS
摘要 The invention relates to compounds of the formula (I), wherein R1, R2, X and Y have the meaning specified in claim 1, are inhibitors of TBK1 and IotaKappaKappaepsilon, and can be used, inter alia, for the treatment of cancer and inflammatory diseases.
申请公布号 WO2013034238(A1) 申请公布日期 2013.03.14
申请号 WO2012EP03449 申请日期 2012.08.13
申请人 MERCK PATENT GMBH;HOELZEMANN, GUENTER;DORSCH, DIETER;EGGENWEILER, HANS-MICHAEL 发明人 HOELZEMANN, GUENTER;DORSCH, DIETER;EGGENWEILER, HANS-MICHAEL
分类号 C07D401/12;A61K31/4433;A61K31/506;C07D401/14;C07D405/14;C07D413/14;C07D417/14;C07D471/04;C07D491/10 主分类号 C07D401/12
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