发明名称 Phosphonic acid compounds as inhibitors of serine proteases
摘要 The present invention is directed to phosphonic acid compounds useful as serine protease inhibitors, compositions thereof and methods for treating inflammatory and serine protease mediated disorders.
申请公布号 US8394804(B2) 申请公布日期 2013.03.12
申请号 US20080288920 申请日期 2008.10.24
申请人 GRECO MICHAEL N.;ALMOND, JR. HAROLD R.;DE GARAVILLA LAWRENCE;HAWKINS MICHAEL J.;HUMORA MICHAEL J.;QIAN YUN;WALKER DONALD GILMORE;CESCO-CANCIAN SERGIO;NILSEN CHRISTOPHER NORMAN;PATEL MITUL N.;SORGI KIRK LEONERD;POWELL EUGENE;JANSSEN PHARMACEUTICA N.V. 发明人 GRECO MICHAEL N.;ALMOND, JR. HAROLD R.;DE GARAVILLA LAWRENCE;HAWKINS MICHAEL J.;HUMORA MICHAEL J.;QIAN YUN;WALKER DONALD GILMORE;CESCO-CANCIAN SERGIO;NILSEN CHRISTOPHER NORMAN;PATEL MITUL N.;SORGI KIRK LEONERD;POWELL EUGENE
分类号 A61K31/4965;C07D241/04;C07D295/00;C07F9/38;C07F9/572;C07F9/59;C07F9/6509;C07F9/655;C07F9/6558;C07F9/6561 主分类号 A61K31/4965
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