发明名称 CRYSTAL OF DI(ARYLAMINO)ARYL COMPOUND
摘要 Provided are crystals of compound A which have properties suitable for industrial production. MEANS FOR SOLVING As the results of intensive studies to provide crystals of compound A having an inhibitory activity on the kinase activity of an EML4-ALK fusion protein and a mutant EGFR protein, crystals of compound A were found. Moreover, it was found that A04-type crystal of compound A, from among the aforesaid crystals of compound A, unexpectedly have preferred properties as a drug substance.
申请公布号 US2013059855(A1) 申请公布日期 2013.03.07
申请号 US201113698183 申请日期 2011.05.16
申请人 SHIMADA ITSURO;HIRAKURA YUTAKA;YAMAZAKI KOUJI;TAKEGUCHI KAZUHIRO;UEDA NORIHIRO;ASTELLAS PHARMA INC. 发明人 SHIMADA ITSURO;HIRAKURA YUTAKA;YAMAZAKI KOUJI;TAKEGUCHI KAZUHIRO;UEDA NORIHIRO
分类号 A61K31/53;A61P35/00;C07D401/14 主分类号 A61K31/53
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