| 摘要 |
Disclosed are intermediate compounds for use in the synthesis of compounds of Formula 1, including all geometric and stereoisomers, N-oxides, and salts thereof,
wherein
J
is a phenyl optionally substituted with one to four substituents independently selected from R 5 ; or J is a heterocyclic ring selected from the group consisting of J-1 to J-8;
R 4
is C 4 -C 12 alkylcycloalkyl, C 5 -C 12 alkenylcycloalkyl, C 5 -C 12 alkynylcycloalkyl, C 4 -C 12 cycloalkylalkyl, C 5 -C 12 cycloalkylalkenyl, C 5 -C 12 cycloalkylalkynyl, C 4 -C 12 cycloalkenylalkyl or C 4 -C 12 alkylcycloalkenyl; each optionally substituted with one to six substituents selected from CH 3 and halogen; or
R 4
is C 3 -C 5 oxiranylalkyl, C 3 -C 5 thiiranylalkyl, C 4 -C 6 oxetanylalkyl, C 4 -C 6 thietanylalkyl, 3-oxetanyl or 3-thietanyl, each optionally substituted with one to five substituents independently selected from C 1 -C 3 alkyl, C 1 -C 3 haloalkyl, halogen, CN, C 2 -C 4 alkoxycarbonyl and C 2 -C 4 haloalkoxycarbonyl; or
R 4
is C 3 -C 5 aziridinylalkyl, C 4 -C 6 azetidinylalkyl or 3-azetidinyl, each with R 10 attached to the nitrogen atom, and optionally substituted on carbon atoms with one to five substituents independently selected from C 1 -C 3 alkyl, C 1 -C 3 haloalkyl, halogen, CN, C 2 -C 4 alkoxycarbonyl and C 2 -C 4 haloalkoxycarbonyl; and
R 1a R 1b R 2 R 3 and R 5
are as defined in the disclosure. |
