| 摘要 |
THIS INVENTION RELATES TO PROCESSES FOR THE PRODUCTION OF OPTICALLY ACTIVE 2-(DISUBSTITUTED ARYL) CYCLOPROPYLAMINE COMPOUNDS AND OPTICALLY ACTIVE 2-(DISUBSTITUTED ARYL) CYCLOPROPANE CARBOXAMIDE COMPOUNDS WHICH ARE USEFUL INTERMEDIATES FOR THE PREPARATION OF PHARMACEUTICAL AGENTS, AND IN PARTICULAR THE COMPOUND [ 1S-(1?,2? 3?(1S*,2R*),5?)]-3-[7-[2-(3,4-DIFLUOROPHENYL)-CYCLOPROPYL]AMINO]-5-(PROPYLTHIO)-3H-1,2,3-TRIAZOLO[4,5- D]PYRIMIDIN-3-YL)-5-(2-HYDROXYETHOXY)-CYCLOPENTANE-1,2-DIOL. |
